| (3H)-DPCPX A1ARs | (3H)-ZM 241385 A2AARs | (3H)-MRE2029F20 A2BARs | (3H)-MRE3008F20 A3ARs |
---|---|---|---|---|
Healthy controls n = 90 | KD = 1.76 ± 0.08 nM Bmax = 34 ± 2 fmol/mg protein | KD = 1.41 ± 0.10 nM Bmax = 58 ± 4 fmol/mg protein | KD = 2.29 ± 0.14 nM Bmax = 55 ± 3 fmol/mg protein | KD = 1.92 ± 0.09 nM Bmax = 137 ± 9 fmol/mg protein |
ERA patients n = 32 | KD = 1.74 ± 0.06 nM Bmax = 33 ± 2 fmol/mg protein | KD = 2.09 ± 0.14* nM Bmax = 185 ± 12* fmol/mg protein | KD = 2.29 ± 0.10 nM Bmax = 55 ± 2 fmol/mg protein | KD = 3.03 ± 0.14* nM Bmax = 290 ± 15* fmol/mg protein |
RA patients n = 63 | KD = 1.69 ± 0.07 nM Bmax = 35 ± 2 fmol/mg protein | KD = 1.93 ± 0.12* nM Bmax = 195 ± 13* fmol/mg protein | KD = 2.36 ± 0.07 nM Bmax = 54 ± 2 fmol/mg protein | KD = 3.47 ± 0.21* nM Bmax = 328 ± 22* fmol/mg protein |