Cell type | Stimulation | EC 50 in nM (peak concentration, pg/mL) | ||||||
---|---|---|---|---|---|---|---|---|
TNFα | IL-6 | IL-1β | MCP-1 | IL-8 | Histamine | PGD2 | ||
THP-1 |
FcγR LPS |
0.9 (577) > 10,000 (934) |
ND > 10,000 (638) |
5.2 (80) ND |
ND ND | |||
Primary human monocytes |
FcγR LPS |
2.6 (6854) > 10,000 (2100) |
3.9 (1380) > 10,000 (528) |
0.5 (100) ND |
908 (3593) ND | |||
Primary human macrophages Primary mouse macrophages |
FcγR FcγR |
561 (337) 4.9 (126) |
1299 (1500) 0.9 (404) |
26.6 (132) 5.1 (22) |
422 (1451) 183 (676) | |||
RAW 267.4 Primary human macrophages |
FcγR (cFb) FcγR (cFb) |
8.7 (619) 113 (1350) |
ND ND |
ND ND |
ND ND | |||
Human cultured mast cells |
FcεR FcγR |
61 (236) 2.1 (67) |
ND ND |
ND ND |
2.2 (341) ND |
32 (722) 7.7 (263) |
25 (460*) 24 (238*) |
21 (1573) 14 (575) |
* ng/mL |